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Food and Drug Administration placed a box warning on GLP-1 medications due to this risk in rodents

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Gases: Small molecular gases like oxygen and carbon dioxide can freely cross the BBB to meet the brains oxygen demand

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Most patients experience brief discomfort during or immediately after injection that resolves within minutes to hours

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doi: 10.1111/dme.14953 14 BurtonPSmitHJLightowlerHJ

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Retatrutide's glucagon receptor agonism adds an additional layer of heart rate elevation beyond what GLP-1 alone would produce

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